HJC0350CAS号: 885434-70-8分子式: C15H19NO2S分子量: 277.38描述纯度储存/保存方法可溶性/溶解性靶点In vitro(体外研究)参考文献
产品描述 | |
描述 |
HJC0350 is a potent and selective EPAC2 inhibitor with IC50 of 0.3 μM, exhibiting no inhibition on Epac1.
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纯度 |
98%
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储存/保存方法 |
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
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基本信息 | |
可溶性/溶解性 |
DMSO:52 mg/mL warmed (187.46 mM)
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生物活性 | |
靶点 |
EPAC2
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In vitro(体外研究) |
HJC0350 selectively blocks cAMP-induced EPAC2 activation but do not inhibit cAMP-mediated PKA activation. In HEK293/EPAC2-FL cells, HJC0350 also inhibits 007-AM mediated cellular activation of EPAC2.
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参考文献 | |
参考文献 |
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分子结构图