CGP 35348CAS号: 123690-79-9分子式: C8H20NO4P分子量: 225.22描述应用储存/保存方法形态别名密度熔点沸点折射率IC50PK值可溶性/溶解性MDLPubChem CID
产品描述 | |
描述 |
CGP 35348 is a selective GABA (GABAB) receptor antagonist (IC50= 34 μM). CGP 35348 has higher affinity for postsynaptic versus presynaptic receptors.
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应用 |
a selective GABAB receptor antagonist
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储存/保存方法 |
Store at 4° C
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形态 |
Solid
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基本信息 | |
别名 |
(3-Aminopropyl)(diethoxymethyl)phos phinic acid
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密度 |
1.13 g/cm3 (Predicted)
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熔点 |
81.49° C (Predicted)
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沸点 |
400.54° C at 760 mmHg (Predicted)
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折射率 |
n20D 1.46 (Predicted)
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IC50 |
GABA B receptor: IC50 = 2.5 µM (rat); GABAB R1: IC50 = 27 µM (human)
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PK值 |
pKa: 2.02 (Predicted), pKb: 10.19 (Predicted)
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可溶性/溶解性 |
Soluble in water (100 mM).
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MDL |
MFCD00882736
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PubChem CID |
107699
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