AG-183CAS号： 122520-90-5分子式： C13H8N4O3分子量： 268.23描述纯度储存/保存方法形态别名外观密度熔点沸点折射率IC50可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
Tyrphostin 51 is a potent inhibitor of EGFR (EGF receptor) kinase activity (IC50=0.8 μM). Inhibition is mixed competitive with ATP and substrate. |
| 纯度 |
98%
|
| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
|
| 形态 |
Solid
|
| 基本信息 | |
| 别名 |
Tyrphostin A51；Tyrphostin 51
|
| 外观 |
solid
|
| 密度 |
~1.6 g/cm3 (Predicted)
|
| 熔点 |
231.43° C (Predicted)
|
| 沸点 |
~788.2° C at 760 mmHg (Predicted)
|
| 折射率 |
n20D 1.76
|
| IC50 |
EGF receptor kinase: IC50 = 0.8 µM (human epidermoid carcinoma cell line A431)
|
| 可溶性/溶解性 |
Soluble in water (0.5 mg/mL) at 25° C, DMSO:PBS(pH 7.2, 1:1), DMSO (50 mg/mL), DMF, and ethanol.
|
| MDL |
MFCD00133903
|
| PubChem CID |
5328807
|
分子结构图
