UB 165 Fumarate

UB 165 FumarateCAS号: 2454492-43-2分子式: C17H19ClN2O4分子量: 350.8描述纯度储存/保存方法靶点In vitro(体外研究)

产品描述
描述
UB 165 fumarate is an agonist of the nAChR, a partial agonist of the α4β2 subtype, and a full agonist of the α3β2 subtype, with a Ki value of 0.27 nM for binding to [3H]-nicotine measured in rat brain.
纯度
98%
储存/保存方法
Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution.
生物活性
靶点
nicotine in rat brain:0.27 nM(ki), nicotine in rat brain(ki):ki:0.27 nM
In vitro(体外研究)
UB-165 fumarate exhibits an EC50 value of 88 nM for stimulating [3H]-dopamine release from striatal synaptosomes.[1]