SKF 83959CAS号： 80751-85-5分子式： C18H20ClNO2•HBr分子量： 398.73描述应用纯度储存/保存方法形态别名熔点折射率IC50Ki 数据可溶性/溶解性MDLPubChem CID
| 产品描述 | |
| 描述 |
SKF 83959 is a D1DR (D1)-like partial agonist. It may act as an antagonist, exhibiting antiparkinsonian effects and antagonizing the behavioral effects of cocaine. SKF 83959 is an activator of D1DR and D5DR.
|
| 应用 |
A D1-like partial agonist
|
| 纯度 |
≥98%
|
| 储存/保存方法 |
Desiccate at room temperature
|
| 形态 |
Solid
|
| 基本信息 | |
| 别名 |
SKF 83959 HBr; SKF 83959 hydrobromide
|
| 熔点 |
250° C
|
| 折射率 |
n20D ~1.62 (Predicted)
|
| IC50 |
Plasmodium falciparum: IC50 = 7.94 µM
|
| Ki 数据 |
D1 receptor: Ki= 1.18 nM (rat); D5 receptor: Ki= 7.56 nM (rat); D3 receptor: Ki= 399 nM (rat); D2 receptor: Ki= 920 nM (rat)
|
| 可溶性/溶解性 |
Soluble in DMSO (>20 mg/ml). Insoluble in water.
|
| MDL |
MFCD03792727
|
| PubChem CID |
11957685
|