PD 168568 diHydrochlorideCAS号： 1782532-06-2分子式： C22H29Cl2N3O分子量： 422.39描述纯度储存/保存方法可溶性/溶解性靶点In vitro(体外研究)In vivo(体内研究)
| 产品描述 | |
| 描述 |
PD 168568 dihydrochloride is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).
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| 纯度 |
98%
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| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
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| 基本信息 | |
| 可溶性/溶解性 |
DMSO:55 mg/mL (130.21 mM)
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| 生物活性 | |
| 靶点 |
D4 Receptor:8.8 nM (ki)
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| In vitro(体外研究) |
PD 168568 dihydrochloride has good selective for D4 receptor(Ki of 1842 nM for D2 receptor)[1].
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| In vivo(体内研究) |
PD 168568 dihydrochloride inhibit amphetamine stimulated locomotor activity in the rat[1].
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