NSC 663284CAS号： 383907-43-5分子式： C15H16ClN3O3 分子量： 321.76描述纯度储存/保存方法别名外观可溶性/溶解性
| 产品描述 | |
| 描述 |
NSC 663284 (DA-3003-1) is a potent, cell-permeable, and irreversible Cdc25 dual specificity phosphatase inhibitor, has an IC50 for Cdc25B2 of 0.21 μM. NSC 663284 exhibits mixed competitive kinetics against Cdc25A, Cdc25B(2), and Cdc25C with Ki values of 29, 95, and 89 nM, respectively. NSC 663284 inhibits NSD2 (IC50 of 170 nM) through a direct interaction with the catalytic SET domain (Kd of 370 nM).
|
| 纯度 |
98%
|
| 储存/保存方法 |
Store at -20℃ for one year（Powder）；Store at 2-4℃ for two weeks；Store at -20℃ for six months after dissolution.
|
| 基本信息 | |
| 别名 |
DA-3003-1
|
| 外观 |
red solid
|
| 可溶性/溶解性 |
DMSO : ≥ 100 mg/mL (310.79 mM)
|
分子结构图
